2-SUBSTITUTED 5-(HETERO)ALKYL-6-HYDROXYPYRIMIDINE-4(1H)-ONES WITH NOOTROPIC ACTIVITY Russian patent published in 2023 - IPC A61K31/513 A61P25/28 C07D239/66 C07D403/12 C07D417/04 

Abstract RU 2793806 C1

FIELD: pharmaceuticals.

SUBSTANCE: invention relates to pharmaceuticals, namely the use of 2-substituted 5-(hetero)alkyl-6-hydroxypyrimidine-4(1H)-ones of the general formula

,

where R=i-Pr, s-Pen, i-Pen, MeSCH2CH2, R1=SCH2CH2N(CH3)2, SCH2CH2N(CH3СH2)2, SCH2CH2N(СH2)4, SCH2CH2N(СH2)5, SCH2CH2SCH3, thiomorpholin-4-yl, or their hydrochloric acid salts as active cores of medicinal products with nootropic properties.

EFFECT: effective nootropic action.

1 cl, 2 tbl

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RU 2 793 806 C1

Authors

Novakov Ivan Aleksandrovich

Tyurenkov Ivan Nikolaevich

Kovalev Nikolaj Sergeevich

Bakulin Dmitrij Aleksandrovich

Kurkin Denis Vladimirovich

Petrov Vladimir Ivanovich

Shejkin Dmitrij Stanislavovich

Kirillov Ivan Aleksandrovich

Vernigora Andrej Aleksandrovich

Brunilina Lejla Lipparitovna

Navrotskij Maksim Borisovich

Dates

2023-04-06Published

2022-01-14Filed