AZABICYCLIC AND DIAZEPINE DERIVATIVES FOR THE TREATMENT OF OPHTHALMIC DISORDERS Russian patent published in 2023 - IPC C07D471/04 C07D471/08 A61K31/439 A61P27/10 

Abstract RU 2795521 C2

FIELD: organic chemistry.

SUBSTANCE: invention relates to a heterocyclic compound or to a pharmaceutical composition based on the said compound.

EFFECT: effective modulation of muscarinic receptors by the said compound useful for the treatment of ophthalmic diseases.

7 cl, 52 dwg, 1 tbl, 25 ex

Similar patents RU2795521C2

Title Year Author Number
AMINOPYRIDINE DERIVATIVES AND THEIR USE AS SELECTIVE ALK-2 INHIBITORS 2022
  • Li, Jialiang
  • Arista, Luca
  • Babu, Sreehari
  • Bian, Jianwei
  • Cui, Kai
  • Dillon, Michael Patrick
  • Lattmann, Rene
  • Liao, Lv
  • Lizos, Dimitrios
  • Ramos, Rita
  • Stiefl, Nikolaus Johannes
  • Ullrich, Thomas
  • Usselmann, Peggy
  • Wang, Xiaoyang
  • Waykole, Liladhar Murlidhar
  • Weiler, Sven
  • Zhang, Yubo
  • Zhou, Yizong
  • Zhu, Tingying
RU2803084C1
AMINOPYRIDINE DERIVATIVES AND APPLICATION THEREOF AS SELECTIVE ALK-2 INHIBITORS 2017
  • Li, Tszyalyan
  • Arista, Luka
  • Babu, Srikhari
  • Byan, Tszyanvej
  • Tsuj, Kaj
  • Dillon, Majkl Patrik
  • Lattmann, Rene
  • Lyao, Lv
  • Lizos, Dimitrios
  • Ramos, Rita
  • Shtifl, Nikolaus Jokhannes
  • Ullrikh, Tomas
  • Usselmann, Peggi
  • Van, Syaoyan
  • Vajkole, Liladkhar Murlidkhar
  • Vajler, Sven
  • Chzhan, Yujbo
  • Chzhou, Itszun
  • Chzhu, Tinin
RU2777979C2
SPIRO-FUSED PIPERIDINE DERIVATIVES FOR APPLICATION AS INHIBITORS OF EXTERNAL MEDULLAR LAYER POTASSIUM CHANNEL 2013
  • Din Fa-Syan
  • Dun Shuchzhi
  • Fri Dzhessika
  • Gu Sin
  • Tszyan Tszinlun
  • Pasternak Aleksander
  • Tan Khajfyn
  • U. Chzhitsaj
  • Yuj Yan
  • Sudzuki Takao
RU2642066C2
CONDENSED TRICYCLIC BENZIMIDAZOLE DERIVATIVES AS MODULATORS OF TNF ACTIVITY 2014
  • Aleksander Rikki Piter
  • Kalmiano Mark Daniel
  • Defejs Sabine
  • Dyure Veronik
  • Delini Mikhael
  • Kher Yag Paul
  • Dzhekson Viktoriya Elizabet
  • Keje Zhan
  • Kroplin Boris
  • Mak-Koss Malkolm
  • Sabnis Jogesh Anil
  • Selbi Mattyu Dankan
  • Svinnen Dominik Lui Leon
  • Van-Khautvin Natali
  • Chzhu Chzhaonin
  • Vener Folkmar
  • Khajnelt Uve
RU2689777C1
AMINOPYRIDINE DERIVATIVES AND THEIR USE AS SELECTIVE ALK-2 INHIBITORS 2017
  • Li, Jialiang
  • Arista, Luca
  • Babu, Sreehari
  • Bian, Jianwei
  • Cui, Kai
  • Dillon, Michael Patrick
  • Lattmann, Rene
  • Liao, Lv
  • Lizos, Dimitrios
  • Ramos, Rita
  • Stiefl, Nikolaus Johannes
  • Ullrich, Thomas
  • Usselmann, Peggy
  • Wang, Xiaoyang
  • Waykole, Liladhar Murlidhar
  • Weiler, Sven
  • Zhang, Yubo
  • Zhou, Yizong
  • Zhu, Tingying
RU2747318C2
FUSED TRICYCLIC IMIDAZOLE DERIVATIVES AS MODULATORS OF TNF ACTIVITY 2014
  • Aleksander Rikki Piter
  • Brejs Garet Nil
  • Braun Dzhulien Alister
  • Kalmiano Mark Daniel
  • Chovatiya Praful Tulshi
  • Delini Mikhael
  • Gallimor Ellen Oliviya
  • Kher Yag Paul
  • Dzhekson Viktoriya Elizabet
  • Kroplin Boris
  • Mak-Koss Malkolm
  • Kuinsi Dzhoanna Rejchel
  • Sabnis Jogesh Anil
  • Svinnen Dominik Lui Leon
  • Chzhu Chzhaonin
  • Khajnelt Uve
  • Vener Folkmar
RU2679914C9
HETEROCYCLIC COMPOUNDS AND USE THEREOF FOR PREVENTING OR TREATING BACTERIAL INFECTIONS 2016
  • Brias, Julie
  • Caravano, Audrey
  • Chasset, Sophie
  • Chevreuil, Francis
  • Faivre, Fabien
  • Ledoussal, Benoit
  • Le Strat, Frederic
  • Richard, Sebastien
  • Simon, Christophe
  • Vomscheid, Sophie
RU2715058C2
MACROCYCLIC COMPOUNDS AS STING AGONISTS AND METHODS USING THEM AND WAYS OF USE THEREOF 2020
  • Karche, Navnath Popat
  • Banerjee, Moloy
  • Gupta, Nishant Ramnivasji
  • Jadhav, Ganesh Rajaram
  • Vyavahare, Vinod Popatrao
  • Das, Amit Kumar
  • Walke, Deepak Sahebrao
  • Kalhapure, Vaibhav Madhukar
  • Bhoskar, Smita Aditya
  • Ramdas, Vidya
  • Palle, Venkata P.
  • Kamboj, Rajender Kumar
RU2825271C2
CONDENSED DERIVATIVES OF IMIDAZOLE AND PYRAZOLE AS MODULATORS OF ACTIVITY TNF 2014
  • Braun Dzhulien Alister
  • Kalmiano Mark Daniel
  • Dzhouns Elizabet Perl
  • Kroplin Boris
  • Ryuberson Dzhejms Tomas
  • Selbi Mattyu Dankan
  • Sho Majkl Alan
  • Chzhu Chzhaonin
RU2686117C1
SUBSTITUTED 3-AZABICYCLO[3_1_0]HEXANES AS KETOHEXOKINASE INHIBITORS 2016
  • Dowling, Matthew
  • Fernando, Dilinie
  • Futatsugi, Kentaro
  • Huard, Kim
  • Magee, Thomas Victor
  • Raymer, Brian
  • Shavnya, Andre
  • Smith, Aaron
  • Thuma, Benjamin
  • Tsai, Andy
  • Tu, Meihua
RU2696269C1

RU 2 795 521 C2

Authors

Ellis, David

Ketelson, Howard Allen

Dates

2023-05-04Published

2018-11-02Filed