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(19)

(11)

2 809 022

(13)

(51)

IPC

C07D403/04(2006-01-01)

C07D403/14(2006-01-01)

C07D401/14(2006-01-01)

C07D405/14(2006-01-01)

A61K31/505(2006-01-01)

A61K31/4375(2006-01-01)

A61K31/5355(2006-01-01)

A61P35/00(2006-01-01)

(21) (22)

Application

2020130864, 2019-02-21

(24)

Start date

2019-02-21

(22)

Actual filing date

2019-02-21

(45)

Published

2023-12-06

(72)

Inventor

Lejrson, Lyuk, L.Chin, Emili, N.Chatterdzhi, ArnabKumar, ManozhAlbero, Ana, Mariya, GamoPetrassi, MajkShults, PiterYu, ChenguangTamijya, DzhunkoVerne, UilyamGupta, AnilModukuri, Ramkumar

(73)

Holder

Ze Skripps Riserch Instityut

AGONISTS OF STING INTERFERON GENE STIMULATOR Russian patent published in 2023 - IPC C07D403/04 C07D403/14 C07D401/14 C07D405/14 A61K31/505 A61K31/4375 A61K31/5355 A61P35/00

Abstract RU 2809022 C2

FIELD: gene engineering.

SUBSTANCE: invention relates to a group of compounds represented by structural formulas in claim 1 with agonistic biological activity of the stimulator of interferon genes (STING) that can find their use in medicine in the treatment of tumors in patients suffering from them.

EFFECT: obtaining agonists of sting interferon gene stimulator.

3 cl, 3 dwg, 3 tbl, 2 ex

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RU 2 809 022 C2

Authors

Lejrson, Lyuk, L.

Chin, Emili, N.

Chatterdzhi, Arnab

Kumar, Manozh

Albero, Ana, Mariya, Gamo

Petrassi, Majk

Shults, Piter

Yu, Chenguang

Tamijya, Dzhunko

Verne, Uilyam

Gupta, Anil

Modukuri, Ramkumar

Dates

2023-12-06—Published

2019-02-21—Filed