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(19)

(11)

2 813 691

(13)

(51)

IPC

C07D213/82(2006-01-01)

C07D237/24(2006-01-01)

C07D239/28(2006-01-01)

C07D401/04(2006-01-01)

C07D403/04(2006-01-01)

C07D413/04(2006-01-01)

C07D417/04(2006-01-01)

A61K31/4418(2006-01-01)

A61K31/501(2006-01-01)

A61K31/506(2006-01-01)

A61P35/00(2006-01-01)

(21) (22)

Application

2022107208, 2020-08-21

(24)

Start date

2020-08-21

(22)

Actual filing date

2020-08-21

(45)

Published

2024-02-15

(72)

Inventor

Petrassi, Khenk Majkl DzhejmsYuj, ChenianVan, TszeChatterdzhi, Arnab K.Albero, Ana Mariya GamoGupta, AnilTamijya, DzhankoShults, Piter Dzh.Dzhonson, KristenChu, AlanChin, EmiliLejrson, Lyuk L.

(73)

Holder

Ze Skripps Riserch Instityut

BICYCLIC AGONISTS OF STING INTERFERON GENE STIMULATOR Russian patent published in 2024 - IPC C07D213/82 C07D237/24 C07D239/28 C07D401/04 C07D403/04 C07D413/04 C07D417/04 A61K31/4418 A61K31/501 A61K31/506 A61P35/00

Abstract RU 2813691 C2

FIELD: pharmaceuticals.

SUBSTANCE: invention relates to chemical compounds and their pharmaceutically acceptable salts given in the claims. The invention also relates to a method of treating a tumor, a pharmaceutical composition and the use of compounds or their pharmaceutically acceptable salts according to the invention for treating a tumor.

EFFECT: using a compound as an agonist of interferon genes stimulator (STING) in the treatment of tumors.

6 cl, 3 tbl, 3 ex

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RU 2 813 691 C2

Authors

Petrassi, Khenk Majkl Dzhejms

Yuj, Chenian

Van, Tsze

Chatterdzhi, Arnab K.

Albero, Ana Mariya Gamo

Gupta, Anil

Tamijya, Dzhanko

Shults, Piter Dzh.

Dzhonson, Kristen

Chu, Alan

Chin, Emili

Lejrson, Lyuk L.

Dates

2024-02-15—Published

2020-08-21—Filed