PYRIDINONE COMPOUNDS AS SELECTIVE CYTOTOXIC AGENTS AGAINST HIV-INFECTED CELLS Russian patent published in 2024 - IPC C07D401/06 C07D403/06 A61K31/4412 A61P31/18 

Abstract RU 2816090 C2

FIELD: medicine; pharmaceutics.

SUBSTANCE: invention relates to pyridinone derivatives of formula I or a pharmaceutically acceptable salt thereof and pharmaceutical compositions based thereon, having cell killing activity, activated by small molecules (SMACK), and having activity for selective destruction of HIV-infected cells expressing GAG-POL.

EFFECT: using the invention enables treating HIV infections, as well as treating and preventing or delaying the onset or progression of AIDS or AIDS-associated complex (ARC).

16 cl, 16 tbl, 43 ex

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RU 2 816 090 C2

Authors

Converso, Antonella

El Marrouni, Abdellatif

Forster, Ashley

Frie, Jessica, L.

Hunter, David, N.

Wang, Cheng

Wang, Deping

Dates

2024-03-26Published

2020-05-18Filed