Patenton — panteon of patents

(19)

RU

(11)

2 817 349

(13)

C1

(51)

IPC

C07D487/08(2006-01-01)

A61K31/4995(2006-01-01)

A61P35/00(2006-01-01)

A61P19/02(2006-01-01)

A61P29/00(2006-01-01)

A61P25/28(2006-01-01)

A61P37/00(2006-01-01)

A61P31/04(2006-01-01)

A61P31/14(2006-01-01)

(21) (22)

Application

2022135100, 2021-06-30

(24)

Start date

2021-06-30

(22)

Actual filing date

2021-06-30

(45)

Published

2024-04-15

(72)

Inventor

Gerstenberger, Brajan StefenTszyao, VenkhuaLall, Mandzhinder SingkhLira, RikardoShnute, Mark Edvard

(73)

Holder

Pfajzer Ink.

AMINOPYRIMIDINYL DERIVATIVES Russian patent published in 2024 - IPC C07D487/08 A61K31/4995 A61P35/00 A61P19/02 A61P29/00 A61P25/28 A61P37/00 A61P31/04 A61P31/14 

Abstract RU 2817349 C1

FIELD: medicine; pharmaceutics.

SUBSTANCE: invention relates to compounds of formulas IA, IB, IC, ID or to their pharmaceutically acceptable salts. Invention also relates to a pharmaceutical composition, a pharmaceutical combination, and a method of treating or preventing a disease or pathological condition for which a JAK1 inhibitor is indicated, based on said compounds.

EFFECT: obtaining novel compounds which can be used in medicine as medicinal agents for treating diseases for which a JAK1 inhibitor is indicated.

17 cl, 2 dwg, 5 tbl, 4 ex

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RU 2 817 349 C1

Authors

Gerstenberger, Brajan Stefen

Tszyao, Venkhua

Lall, Mandzhinder Singkh

Lira, Rikardo

Shnute, Mark Edvard

Dates

2024-04-15—Published

2021-06-30—Filed

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