BORYLATED AMINO ACID COMPOSITIONS FOR USE IN BORON NEUTRON CAPTURE THERAPY AND METHODS THEREOF Russian patent published in 2024 - IPC A61K31/69 A61P35/00 C07F5/02 

Abstract RU 2818817 C2

FIELD: chemistry.

SUBSTANCE: invention relates to a composition for use in boron-neutron capture therapy containing borylated amino acids. Borylated amino acids have the following chemical structure:

where E = CONHB12H11 and X=H. Also disclosed are kits and standard dosage forms containing said composition.

EFFECT: disclosed composition can be administered to patients as a neutron capture agent to provide a method of treating cancer, immunological disorders and other diseases using a boron-neutron capture therapy agent.

8 cl, 14 dwg, 1 tbl, 13 ex

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RU 2 818 817 C2

Authors

Torgov, Michael, Y.

Martin, Tioga, J.

Raitano, Arthur, B.

Dates

2024-05-06Published

2020-03-04Filed