FIELD: medicine, pharmaceutics.
SUBSTANCE: invention refers to a compound of formula (I) where one of R1 and R2 represents -NH-X-Y-Z, and another represents -OH; where X represents -(CH2)m- where m is equal to 0, 1, 2, 3 or 4; Y represents carborane where at least one boron atom represents 10B; and Z represents H; and its pharmaceutically acceptable salts, solvates and stereoisomers. Also, the pharmaceutical compositions, application of the compound of formula (I) and a method of producing the compound of formula (I) are offered.
EFFECT: production of the compounds effective for boron neutron capture therapy.
15 cl, 6 ex, 3 tbl
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Authors
Dates
2011-07-10—Published
2006-08-17—Filed