BENZOXAZINONE COMPOUNDS AS DOUBLE INHIBITORS KLK5/7 Russian patent published in 2024 - IPC C07D498/04 A61K31/536 A61P17/00 

Abstract RU 2831430 C1

FIELD: pharmaceutics.

SUBSTANCE: invention relates to a compound of formula (I), where R is hydrogen, and a pharmaceutical composition thereof for treating a skin disease associated with proteolytic activity of one or more KLK proteases.

EFFECT: disclosed are benzoxazinone compounds as double inhibitors of KLK5/7.

22 cl, 4 dwg, 3 tbl, 6 ex

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RU 2 831 430 C1

Authors

Betz, Andreas

Zamboni, Robert

Dates

2024-12-06Published

2020-09-30Filed