METHOD OF SYNTHESIS OF AZETIDINE DERIVATIVE OR ITS PHARMACEUTICAL ACCEPTABLE SALT Russian patent published in 1995 - IPC

Abstract RU 2048469 C1

FIELD: organic chemistry. SUBSTANCE: product: azetidine derivative of the formula (I) with definite radical values. Reagent 1: compound of the formula (I) where R3-H. Reagent 2: compound of the formula R3-X, where R3 as indicated above, X halogen atom. Reaction conditions: conversion of the group R3 if necessary to any other meaning of the group R3. Synthesized compounds were used as antiallergic and antiasthmatic drugs. EFFECT: improved method of synthesis. 2 tbl

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RU 2 048 469 C1

Authors

Khirosi Fukumi[Jp]

Tosiaki Sakamoto[Jp]

Mitsuo Sugijami[Jp]

Esio Iizuka[Jp]

Takesi Jamaguti[Jp]

Dates

1995-11-20Published

1990-10-04Filed