METHOD OF SYNTHESIS OF DERIVATIVES OF BACCATIN-III OR 10-DESACETYL-BACCATIN-III AND A METHOD OF TAXANE DERIVATIVES SYNTHESIS Russian patent published in 1997 - IPC

Abstract RU 2088578 C1

FIELD: organic chemistry, natural compounds. SUBSTANCE: invention relates to method of synthesis of taxane derivative of the general formula (I) and the use of the synthesized compound for synthesis of taxane derivatives of the general formula (II) . In general formula (I) radical R₁ is acetyl or protecting group, G₁ - protecting group and R - tert. -butoxy radical or phenyl. In general formula (II) R is tert.-butoxy radical or phenyl and R′1

- hydrogen atom or acetyl. EFFECT: improved method of synthesis. 6 cl

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RU 2 088 578 C1

Authors

Ogjusten Ittenzher[Fr]

Dates

1997-08-27—Published

1992-07-08—Filed