DERIVATIVES OF PIPERAZINYLPENTAMIDE AND PHARMACEUTICAL COMPOSITION FOR INHIBITION OF HIV-PROTEASE ACTIVITY Russian patent published in 1999 - IPC

Abstract RU 2131416 C1

FIELD: organic chemistry, medicine, pharmacy. SUBSTANCE: invention relates to new derivatives of piperazinylpentamide of the formula (I) which inhibit activity of protease encoded by human immunodeficiency virus. Invention describes also a pharmaceutical composition based on compound of the formula (I) that is used for inhibition of HIV-infection. EFFECT: enhanced effectiveness. 13 cl, 4 tbl, 17 ex

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RU 2 131 416 C1

Authors

Dzhozef P.Vakka

Brjus D.Dorsi

Dzhejms P.Guar

Katrin M.Khollovej

Rehndell V.Khangejt

Dates

1999-06-10—Published

1992-11-03—Filed