FIELD: organic chemistry, pharmacy. SUBSTANCE: invention describes new substituted 1-naphthylpyrazole-3-carboxamides of the general formula (I) 
where values R, p, n, g, R1-R8,R11-R17,, T are given in p. 1 of the invention claim. Compounds show the significant affinity to the human receptors of neurotensin. Invention describes also a method of their synthesis, a pharmaceutical composition containing these compounds and intermediate compounds of the synthesis. EFFECT: improved method of synthesis, new compounds indicated above, valuable pharmacological properties. 9 cl, 2 tbl, 40 ex
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Year |
Author |
Number |
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1996 |
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1994 |
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1995 |
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1995 |
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|
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1996 |
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|
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1996 |
- Bart Fransis
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