FIELD: organic chemistry, pharmacy. SUBSTANCE: invention relates to N-piperidino-5-(4-chlorophenyl)-1-(2,4-dichloro-phenyl)-4-methylpyrazole-3-carboxamide synthesized by treatment of the compound of the formula (I) 
with 1-aminopiperidine in an organic solvent in the presence of the base. The synthesized compound shows an antagonistic activity with respect to cannabinoid receptors of the central nervous system. EFFECT: improved method of synthesis, valuable pharmacological properties. 10 cl, 1 dwg, 9 ex
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