FIELD: medicine. SUBSTANCE: 4- amino-3-acylquinoline derivatives of general formula I: 
wherein R1 and R3 are C1-6 alkyl; R2 is C1-6 alkyl, halogen, C1-6 alkoxy; R4 is H, C1-6 alkyl, halogen or OH, m is 2 or 3, n is integer of 0,1,2 or pharmaceutically acceptable salts thereof exogenically or endogenically inhibit stimulated secretion of gastric acid are useful for prophylaxis and treatment of inflammatory gastrointestinal diseases. EFFECT: improved properties of the pharmaceutical agent. 13 cl, 57 ex, 1 tbl
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Year |
Author |
Number |
| DERIVATIVES OF IMIDAZO[1,2-A]PYRIDINE, METHODS OF THEIR SYNTHESIS, PHARMACEUTICAL PREPARATION BASED ON THEREOF, METHOD OF INHIBITION OF GASTRIC ACID SECRETION, METHOD OF TREATMENT OF GASTROENTERIC INFLAMMATORY DISEASES AND METHOD OF TREATMENT OF STATES WITH HELICOBACTER PYLORI INFECTION |
1998 |
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- Starke Ingemar
|
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1996 |
- Gustafsson David
- Njustrem Jan-Ehrik
|
RU2176645C2 |
| THROMBIN INHIBITOR-CONTAINING AQUEOUS SOLUTION FOR NONPARENTERAL ADMINISTRATION SHOWING STABILITY AT STORAGE |
1995 |
- Ulla St'Ernfel'T
- Mats Sundgren
|
RU2164803C2 |
| PHENYLETHYL- AND PHENYLPROPYLAMINE COMPOUNDS, METHOD OF THEIR SYNTHESIS AND PHARMACEUTICAL PREPARATION |
1994 |
- Stefan Bengtsson
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RU2133735C1 |
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1997 |
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|
RU2184113C2 |
| DIHYDROPYRIDINES, METHOD OF THEIR SYNTHESIS, PHARMACEUTICAL COMPOSITION BASED ON SAID AND METHOD OF BLOOD PRESSURE DECREASE |
1994 |
- Chell' Jal'Mar Andersson
- Margareta Nordlander
- Rol'F Krister Vesterlund
|
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| DERIVATIVES OF (1-PHENYL-1-HETEROCYCLYL)ALKANE, METHOD OF THEIR SYNTHESIS, PHARMACEUTICAL PREPARATION SHOWING NEUROPROTECTIVE EFFECT IN BRAIN ISCHEMIA, METHOD OF TREATMENT OF PATIENTS WITH HYPOXIC AND ASPHYXIC BRAIN DAMAGES |
1994 |
- Bernard Robin Bor
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- Alfred Richard Grin
|
RU2137763C1 |
| BICYCLIC DERIVATIVES OF ISOTHIOUREA, METHOD OF THEIR SYNTHESIS AND PHARMACEUTICAL COMPOSITION BASED ON THEREOF |
1996 |
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RU2157802C2 |
| PEPTIDE DERIVATIVES, THEIR STEREOISOMERS OR PHYSIOLOGICALLY ACCEPTABLE SALTS SHOWING ANTITHROMBOSIS, ANTICOAGULATING OR ANTI-INFLAMMATORY ACTIVITY, METHOD OF THEIR SYNTHESIS, PHARMACEUTICAL COMPOSITION, METHOD OF SUPPRESSION OF THROMBIN ACTIVITY, METHOD OF INHIBITION OF KININOGENASES ACTIVITY, USE OF COMPOUNDS AS PARENT SUBSTANCES FOR SYNTHESIS OF THROMBIN INHIBITOR |
1994 |
- Karl Tomas Antonsson
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|
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| DERIVATIVE OF (1-HETEROAZOLYL-1-HETEROCYCLE)-ALKANE OR ITS HEOMETRIC OR OPTIC ISOMERS OR RACEMATES OR ITS PHARMACEUTICALLY ACCEPTABLE ACID SALTS OR ITS SOLVATES, METHODS OF ITS SYNTHESIS, ACYL-SUBSTITUTED COMPOUNDS, PHARMACEUTICAL COMPOSITION SHOWING NEUROPROTECTIVE PROPERTY |
1994 |
- Bernard Robin Bor
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RU2124011C1 |
