DERIVATIVES OF OXAZOLIDINEDIONE, THEIR SYNTHESIS (VARIANTS) AND PHARMACEUTICAL COMPOSITION Russian patent published in 2000 - IPC

Abstract RU 2144030 C1

FIELD: organic chemistry, pharmacy. SUBSTANCE: invention relates to derivatives of oxazolidinedione of the formula: where R means optionally substituted hydrocarbon residue or heterocyclic group; Y means the group as -CO-, -CH(OH) or NR3 where R3 means optionally substituted alkyl group; m = 0 or 1; n = 0, 1 or 2; A means bivalent C1-7-aliphatic hydrocarbon group; R1 means hydrogen atom or alkyl group; ring E means benzene ring having 1 or 2 substituents; L and M mean hydrogen atom, respectively, or L and M can be fused and form the bond at condition that the group is not the group where R2 means alkyl group, or their salts. Compounds decrease blood glucose and lipids content effectively. EFFECT: improved method of synthesis, enhanced effectiveness of compounds. 25 cl, 8 tbl, 114 ex

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RU 2 144 030 C1

Authors

Takasi Sokhda

Khirojuki Odaka

Jju Momoze

Mitsuru Kavada

Dates

2000-01-10Published

1995-11-01Filed