FIELD: organic chemistry, pharmacy. SUBSTANCE: invention describes novel derivatives of phenylamidine of the general formula (I) 
where R means hydrogen atom, alkyl with 1 or 2 carbon atoms or cyclohexyl; Y means 1,4-piperidyl, their tautomers and stereoisomers including their mixtures and salts that can act as an active substance of pharmaceutical composition showing antithrombotic and antiaggregative effect. Invention describes pharmaceutical composition based on the formula (I) also. EFFECT: new compounds indicated above, valuable medicinal properties. 2 cl, 1 tbl
| Title |
Year |
Author |
Number |
| DERIVATIVES OF PYRIDINE, THEIR ENANTIOMERS, CIS- OR TRANS-ISOMERS AND THEIR SALTS AND PHARMACEUTICAL COMPOSITION |
1992 |
- Rajner Zojka
- Tomas Mjuller
- Iogannes Vejzenberger
|
RU2119915C1 |
| CYCLIC NITROGEN-CONTAINING DERIVATIVES, MIXTURE OF THEIR ISOMERS, INDIVIDUAL ISOMERS OR THEIR SALTS |
1994 |
- Frank Khimmel'Sbakh
- Khel'Mut Piper
- Fol'Kkhard Austel'
- Gjunter Lints
- Brajen Gas
- Tomas Mjuller
- Iogannes Vejzenberger
|
RU2126002C1 |
| DIAZEPINONE DERIVATIVES, METHODS OF THEIR SYNTHESIS AND PHARMACEUTICAL COMPOSITION |
1992 |
- Vol'Fgang Ehberlajn[De]
- Gerkhard Mim[De]
- Vol'Fkhard Ehngel'[De]
- Klaus Rudol'F[De]
- Khengi Duds[Nl]
- Kharal'D Tsigler[At]
- Mikhaehl' Ehnttserot[De]
|
RU2081870C1 |
| DERIVATIVES OF PYRIDYL, MIXTURE OF THEIR ISOMERS, OR INDIVIDUAL ISOMERS, OR THEIR PHYSIOLOGICALLY TOLERATED ADDITIVE SALTS SHOWING BIOLOGICAL ACTIVITY |
1991 |
- Rajner Zojka[De]
- Vol'Fgang Ehjzert[De]
- Tomas Mjuller[De]
- Iogannes Vejzenberg[De]
|
RU2028292C1 |
| DERIVATIVES OF BENZIMIDAZOLE AND THEIR SALTS AND PHARMACEUTICAL COMPOSITION BASED ON SAID SHOWING ANTAGONISTIC ACTIVITY WITH RESPECT TO ANGIOTENSIN |
1995 |
- Gerkhard Mim
- Norbert Khauel'
- Uve Ris
- Jakobus Konstantinus Antonius Fan Meel'
- Vol'Fgang Vinen
- Mikhaehl' Ehnttserot
|
RU2139869C1 |
| BENZIMIDAZOLE DERIVATIVES AND PHARMACEUTICAL COMPOSITION SHOWING ANTAGONISTIC ACTIVITY WITH RELATION TO ANGIOTENSIN BASED ON THEREOF |
1992 |
- Norbert Khauel'[De]
- Bertkhol'D Narr[De]
- Uve Ris[De]
- Zhak Fan Meel'[De]
- Vol'Fgang Vinen[De]
- Mikhael' Ehnttserot[De]
|
RU2053229C1 |
| ARYLSULFONEAMIDE DERIVATIVES, MIXTURES OF THEIR ISOMERS OR INDIVIDUAL ISOMERS AND THEIR PHYSIOLOGICALLY TOLERANTABLE ADDITIVE SALTS WITH BASES AND PHARMACEUTICAL COMPOSITION SHOWING ANTITHROMBIC ACTIVITY |
1992 |
- Khekel' Armin[Gb]
- Nikl' Jozef[Gb]
- Zojka Rajner[Gb]
- Ajzert Vol'Fgang[Gb]
- Mjuller Tomas[Gb]
- Vajzenberger Jokhannes[Gb]
- Mid Kristofer[Gb]
- Muatsevich Gojko[De]
|
RU2096405C1 |
| FUSED 5-MEMBER HETEROCYCLES OR THEIR SALTS SHOWING ACTIVITY BY AGGREGATION INHIBITION |
1992 |
- Fol'Kkhard Austel'[De]
- Khel'Mut Piper[De]
- Frank Khimmel'Sbakh[De]
- Gjunter Lints[De]
- Tomas Mjuller[De]
- Iokhannes Vajzenberger[De]
- Ehl'Ke Zeeval'Dt-Beker[De]
|
RU2041211C1 |
| (-S)(+)-2- ETHOXY-4- -N-[1-2 (2-PIPERIDINOPHENYL) -3- METHYL -1-BUTYL] -AMINOCARBONYLMETHYL -BEN- ZOIC ACID OR ITS HYDRATE, OR PHARMACEUTICALLY ACCEPTABLE SALT POSSESSING OF GLUCOPENIC ACTION |
0 |
- Volfgang Grell
- Andreas Grajshel
- Gabriele Tsan
- Mikhael Mark
- Khanserg Knorr
- Ekkhard Rupprekht
- Ulrikh Myuller
|
SU1831481A3 |
| DERIVATIVES OF DIPYRIDO-DIAZEPINE AND THEIR PHARMACOLOGICALLY TOLERATED SALTS SHOWING BIOLOGICAL ACTIVITY |
1992 |
- Gjunter Shmidt[De]
- Vol'Fkhard Ehngel[De]
- Gjunter Trummlitts[De]
- Vol'Fgang Ehberlajn[De]
- Karl Khargrejv[Us]
|
RU2024522C1 |
