DERIVATIVES OF PIPERIDINE AND PHARMACEUTICAL PREPARATION BASED ON THEREOF Russian patent published in 2002 - IPC

Abstract RU 2183624 C2

FIELD: organic chemistry, heterocyclic compounds, pharmacy. SUBSTANCE: invention relates to novel derivatives of piperidine of the formula (I) where R1 means benzothienyl, benzofuranyl, naphthyl that can be substituted with halogen atom, C1-C6--alkyl, C1-C6-alkoxy- group; substituted thienyl or substituted furanyl that are substituted with halogen atom, C1-C6-alkyl, C3-C6- cycloalkyl or C1-C6-alkenyl; R2 means halogen atom; R3 means C1-C6-alkyl or C3-C6-cycloalkylmethyl or their pharmaceutically acceptable salts or solvates. Compounds of the formula (I) show an antipsychotic activity and can be used in medicine. EFFECT: new compounds indicated above, valuable medicinal property. 8 cl, 2 tbl

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RU 2 183 624 C2

Authors

Rae Dankan Robertson

Gibson Samuehl Dzhordzh

Dates

2002-06-20Published

1997-11-12Filed