5,5-DISUBSTITUTED 2-METHYL-9,9-DIOXO-9-THIABICYCLO-[4,3,0]NONANES Russian patent published in 2002 - IPC

Abstract RU 2184732 C1

FIELD: organic chemistry of heterocyclic compounds of sulfur. SUBSTANCE: invention relates to thiabicyclic derivatives of the formula (I) showing an antidepressant activity where: R is H, Na, Me, CH₂=CHCH₂,CH₂Ph or CH₃CH₂CH₂CH₂; X is CONH₂,NH₂•HCl, NHBoc, CH₂NH₂ or C(OEt)₂NH₂•HCl. Compounds show low toxicity and the more expressed and stable effect in some tests as compared with standard antidepressants and can be synthesized from available and inexpensive raw. EFFECT: improved valuable medicinal properties of compounds. 2 cl, 3 tbl, 11 ex

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RU 2 184 732 C1

Authors

Shul'Ts Eh.Eh.

Tolstikov G.A.

Sorokina I.V.

Tolstikova T.G.

Dates

2002-07-10—Published

2001-04-26—Filed