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Application

2003118101/04, 2003-06-16

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Start date

2003-06-16

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Actual filing date

2003-06-16

(45)

Published

2005-05-20

(72)

Inventor

Belanov E.F.Pokrovskij A.G.Sandakhchiev L.S.Bormotov N.I.Kotovskaja S.K.Chupakhin O.N.Charushin V.N.Rusinov V.L.

(73)

Holder

Gosudarstvennyj Nauchnyj Tsentr Virusologii I Biotekhnologii

3-PHENYL-6-R-7-R-1,2,4-BENZOTRIAXINES WITH ANTIVIRAL ACTIVITY Russian patent published in 2005 - IPC

Abstract RU 2252218 C2

FIELD: bioactive compounds.

SUBSTANCE: invention relates to new 3-phenyl-1,2,4-benzotriazines and their derivatives of general formula 1

wherein R₁ and R₂are independently fluorine or C₁-C₄-alkoxy, optionally substituted with halogen or tetrahydrofuryl. Compounds of present invention are useful in treatment and prophylaxis of diseases, induced by pathogenic for human and animals viruses including pathogenic for human orthopoxviruses, as well as postvaccinal sequelae.

EFFECT: compounds with improved antiviral activity.

1 cl, 12 ex, 7 tbl

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RU 2 252 218 C2

Authors

Belanov E.F.

Pokrovskij A.G.

Sandakhchiev L.S.

Bormotov N.I.

Kotovskaja S.K.

Chupakhin O.N.

Charushin V.N.

Rusinov V.L.

Dates

2005-05-20—Published

2003-06-16—Filed