COMPOUNDS, PHARMACEUTICAL COMPOSITION AND METHOD FOR INHIBITION OF TUMOR GROWTH (VARIANTS) Russian patent published in 2006 - IPC C07C271/22 A61K31/27 A61P43/00 A61P35/00 

Abstract RU 2276133 C2

FIELD: organic chemistry, medicine, oncology, pharmacy.

SUBSTANCE: invention relates to new compounds of the formula (I) inhibiting tumor growth and angiogenesis wherein each R2 and R3 represents independently hydrogen atom (H), (C1-C4)-alkyl; each X2 and X3 represents independently (C1-C4)-perfluoroalkyl; A represents hydrogen atom (H) or a covalent bond; t represents a whole number 0 or 1 under condition that if A represents hydrogen atom (H) then t = 0, and if A represents a covalent bond then t = 1. Also, invention relates to a pharmaceutical composition and method for inhibition of the tumor growth.

EFFECT: valuable medicinal properties of composition.

32 cl, 3 sch, 5 dwg, 19 ex

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RU 2 276 133 C2

Authors

Boger Dejl L.

Cheresh Dehvid A.

Dates

2006-05-10Published

2001-03-27Filed