BENZOXAZINONE DERIVATIVES AND BASED ON THEM PHARMACEUTICAL COMPOSITION Russian patent published in 2008 - IPC C07D265/36 C07D413/06 C07D291/08 A61K31/538 A61K31/54 A61P25/28

Abstract RU 2328490 C2

FIELD: chemistry.

SUBSTANCE: compounds with the formula are described and its pharmaceutically acceptable salts, where Y, Z, R¹, R², R³, R⁴, R⁵, R⁶, R⁷, R⁸, R⁹, m, n, p and q are as specified in the invention. The obtained compounds have the modulating activity regarding the 5-HT receptors. The pharmaceutical composition which contains the compounds with formula (I) and used in treatment of certain central nervous system diseases is also described.

EFFECT: novel compound group with useful biological properties is obtained.

10 cl, 2 dwg, 7 ex

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RU 2 328 490 C2

Authors

Khans Mag

Mehn Sju

Chukhaj Dzhao

Dates

2008-07-10—Published

2003-11-04—Filed