QUINOLINE DERIVATIVES Russian patent published in 2009 - IPC C07D401/12 A61K31/437 A61P27/02 

Abstract RU 2345991 C2

FIELD: chemistry.

SUBSTANCE: description is given of a compound with general formula Ia , where A and Q each represents H and where the asymmetrical centre in position 3 can be in optically active form, R represents formula Ib and where R1 is an alkyl, containing 1 to 4 carbon atoms, in form of a free base or in form of a pharmaceutical acidic additive salt and a pharmaceutical composition, capable of reducing intraocular pressure, based on this compound. Description is also given of the method of treating glaucoma or myopia and use of formula Ia compound for making medicinal preparations for treating glaucoma and myopia.

EFFECT: new method of treating glaucoma or myopia.

6 cl, 6 ex

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RU 2 345 991 C2

Authors

Gull' Peter

Pombo-Vil'Jar Ehsteban

Dates

2009-02-10Published

2003-03-06Filed