DIAZABICYCLIC ARYL DERIVATIVES USED AS MODULATORS OF CHOLINERGIC RECEPTORS Russian patent published in 2009 - IPC C07D471/08 A61K31/551 A61P25/16 

Abstract RU 2368614 C2

FIELD: medicine.

SUBSTANCE: there described are diazabicyclic aryl derivatives of general formula I , their enantiomers or any mixture of those enantiomers, or their pharmaceutically acceptable salts, where radical values A, L, B and n are given in the description, and pharmaceutical composition containing the above diazabicyclic aryl derivatives.

EFFECT: new compounds represent cholinergic ligands of nicotinic receptors of acetylcholine and modulators of receptors and carrying agents of monoamines, and can be used for treatment of diseases and illnesses related to cholinergic system of central nervous system and periphery nervous system, which are related to activity of muscles, endocrine diseases, inflammatory diseases, and neurodegenerative diseases.

12 cl, 2 ex, 1 tbl

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RU 2 368 614 C2

Authors

Peters Dan

Ol'Sen Gunnar M.

Nil'Sen Ehl'Sebet Ehstergord

Ergensen Tino Djukhring

Timmerman Daniel' B.

Dates

2009-09-27Published

2005-02-01Filed