CYCLOPENTYL DERIVATIVES Russian patent published in 2009 - IPC C07C237/24 A61K31/16 A61P25/00 A61P29/00 A61P13/00 

Abstract RU 2372325 C2

FIELD: chemistry.

SUBSTANCE: formula compound is described, where X is oxygen; R1 is a linear or branched C1-C8-alkyl chain, substituted with phenyl, optionally substituted with halogen atoms; R2, R3 independently represent hydrogen, C1-C3-alkyl chain, halogen, methoxy; R4, R5, R6, R7 independently represent hydrogen, as well as a method of obtaining formula (I) compound, and a pharmaceutical composition.

EFFECT: use of the compound to make a medicinal agent which is effective as a modulator of the sodium and/or calcium channel and, consequently, suitable for preventing, relieving and treating a wide range of pathologies which include neurological, psychiatric, cardiovascular, phlogistic, eye, urological, metabolic and intestinal diseases, where the above mentioned mechanisms are described as playing a pathological role.

6 cl, 11 ex

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Authors

Melloni P'Ero

Sabido David Chibehle Marija

Rehstivo Alessandra

Forlani Roberto

Sal'Vati Patrisija

Dates

2009-11-10Published

2004-11-12Filed