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2 379 306

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IPC

C07D417/14(2006-01-01)

A61K31/541(2006-01-01)

A61K31/549(2006-01-01)

A61P7/02(2006-01-01)

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Application

2008130297/04, 2008-07-22

(24)

Start date

2008-07-22

(22)

Actual filing date

2008-07-22

(45)

Published

2010-01-20

(72)

Inventor

Chupakhin Oleg NikolaevichSidorova Larisa PetrovnaPerova Natal'Ja MikhajlovnaRusinov Vladimir LeonidovichMakarov Vladimir AleksandrovichVasil'Eva Tat'Jana MikhajlovnaVorob'Ev Andrej Ivanovich

(73)

Holder

Gosudarstvennoe Obrazovatel'Noe Uchrezhdenie Vysshego Professional'Nogo Obrazovanija Gosudarstvennyj Tekhnicheskij Universitet-Upi"

2-CYCLOALKYLAMINO-5-THIENYL-1,3,4-THIADIAZINES, HYDROBROMIDES, WITH ANTIAGGREGANT ACTIVITY Russian patent published in 2010 - IPC C07D417/14 A61K31/541 A61K31/549 A61P7/02

Abstract RU 2379306 C1

FIELD: chemistry.

SUBSTANCE: invention relates to organic chemistry and specifically to 2-cycloalkylamino-5-thienyl-1,2,3-thiadiazines hydrobromides with antiaggregant activity , where R=H; CH₃; Br, = morpholino-; thiomorpholino-; pyrrolidino-; 2,6-dimethylmorpholino-; hexamethylenimino-.

EFFECT: obtaining novel compounds which can be used in medicine for treating and preventing such diseases as myocardial infarcation, stroke, rejection of transplanted organs and tissue, and can also prevent embolism and thrombosis formation.

1 cl, 5 tbl, 5 ex

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RU 2 379 306 C1

Authors

Chupakhin Oleg Nikolaevich

Sidorova Larisa Petrovna

Perova Natal'Ja Mikhajlovna

Rusinov Vladimir Leonidovich

Makarov Vladimir Aleksandrovich

Vasil'Eva Tat'Jana Mikhajlovna

Vorob'Ev Andrej Ivanovich

Dates

2010-01-20—Published

2008-07-22—Filed