4-(PHENYLMETHYL AND SUBSTITUTED-PHENYLMETHYL)-IMIDAZOLE-2-THIONIES, ACTING AS SPECIFIC ALPHA-ADRENERGIC AGONISTS Russian patent published in 2010 - IPC C07D233/84 A61K31/4174 

Abstract RU 2383535 C2

FIELD: chemistry.

SUBSTANCE: described are compounds of formula

where R1 independently represents H, alkyl containing 1-4 carbon atoms, p represents an integer selected from 0 and 2, R3 is independently selected from a group consisting of fluoro-substituted alkyl containing 1-4 carbon atoms, F, Cl.

EFFECT: compounds are useful as medicine for mammals, including humans, for treating diseases and relieving conditions which respond to treatment by agonists of alpha2 adrenergic receptors.

12 cl, 1 tbl, 4 ex

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RU 2 383 535 C2

Authors

Khejdelbau Tod M.

Chou Ken

Nguen Fong Kh.

Dzhil Dehniehl V.

Donello Dzhon E.

Garst Majkl E.

Uiler Larri A.

Dates

2010-03-10Published

2005-09-07Filed