NOVEL SALT FORM OF DOPAMINE AGONIST Russian patent published in 2010 - IPC C07D401/04 C07D413/04 A61K31/5377 A61P15/00 

Abstract RU 2393153 C2

FIELD: chemistry.

SUBSTANCE: invention relates to a novel salt form of 5-[(2R,5S)-5-methyl-4-propylmorpholin-2-yl]piridine-2-amine (I): , and specifically to 5-[2R,5S)-5-methyl-4-propylmorpholin-2-yl]pyridine-2-amine di-(1S)-camphorsulphonate (di-S-camsylate), to a pharmaceutical composition having effect on dopamine D3 receptor, as well use of the given compound in preparing a medicinal agent for treating sexual dysfunction and neuropsychiatric disorders and a method of obtaining the said compound and an intermediate compound.

EFFECT: novel salt form of a dopamine agonist which has advantages, specifically is not hygroscopic, has a crystalline form and has high melting point is obtained and described.

11 cl, 9 ex, 2 tbl, 6 dwg

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RU 2 393 153 C2

Authors

Grin Stjuart Piter

Ladzari Oliv'E Alen

Miller Dunkan Charl'Z

Saling Fabris Genri

Dates

2010-06-27Published

2006-01-26Filed