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2 383 549

(13)

C1

(51)

IPC

C07D487/18(2006-01-01)

A61K31/529(2006-01-01)

(21) (22)

Application

2008145611/04, 2008-11-19

(24)

Start date

2008-11-19

(22)

Actual filing date

2008-11-19

(45)

Published

2010-03-10

(72)

Inventor

Denislamova Ekaterina SergeevnaMaslivets Andrej Nikolaevich

(73)

Holder

Gosudarstvennoe Obrazovatel'Noe Uchrezhdenie Vysshego Professional'Nogo Obrazovanija Gosudarstvennyj Universitet"

METHYL 11-ARYL-12-AROYL-9-HYDROXY-4,6-DIMETHYL-3,5,10-TRIOXO-4,6,8,11-TETRAAZATRICYCLO[7,2,1,0]DODEC-2(7)-ENE-1-CARBOXYLATES AND SYNTHESIS METHOD THEREOF Russian patent published in 2010 - IPC C07D487/18 A61K31/529 

Abstract RU 2383549 C1

FIELD: chemistry.

SUBSTANCE: invention relates to organic chemistry, more specifically to novel individual azatricycloeicosanic class compounds. Described are methyl 11-aryl-12-aroyl-9-hydroxy-4,6-dimethyl-3,5,10-trioxo-4,6,8,11-tetraazatricyclo[7.2.1.02,7]dodec-2(7)-ene-1-carboxylates of formula , where Ar1=Ar2=Ph (a), Ar1=C6H4Br-4, Ar2=C6H4Me-4 (b). Also described is a method for synthesis of methyl 11-aryl-12-aroyl-9-hydroxy-4,6-dimethyl-3,5,10-trioxo-4,6,8,11-tetraazatricyclo[7.2.1.02,7]dodec-2(7)-ene-1-carboxylates.

EFFECT: novel compounds are obtained, which can be used as precursors for synthesis of novel heterocyclic systems and in pharmacology.

4 cl, 2 ex

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RU 2 383 549 C1

Authors

Denislamova Ekaterina Sergeevna

Maslivets Andrej Nikolaevich

Dates

2010-03-10—Published

2008-11-19—Filed

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