ALKYL SULPHONAMIDE QUINOLINES WITH AFFINITY TO NK-3 RECEPTORS Russian patent published in 2011 - IPC C07D215/52 A61K31/47 A61P25/18 A61P25/22 A61P25/24 A61P25/28 A61P3/04 A61P35/00 

Abstract RU 2421447 C2

FIELD: chemistry.

SUBSTANCE: compound is ((S)-1-phenyl-propyl)-amide 3-(methane sulphonyl amino)-2-phenyl- quinoline-4-carboxylic acid, stereoisomer, enantiomer or pharmaceutically acceptable salt thereof. The invention also relates to a pharmaceutical composition based on the disclosed compound.

EFFECT: novel derivative of methyl sulphonamide quinoline which can be used to modulate the NK-3 receptor.

2 cl, 10 ex

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RU 2 421 447 C2

Authors

Simpson Tomas

Kang Dzhejms

Ehlbert Dzheffri

Ehlkhambra Kristobal'

Kouiter Dzherard

Vuds Dzhejms

Li Jan

Dates

2011-06-20Published

2006-12-11Filed