AMINOPHOSPHATE DERIVATIVE AND S1P RECEPTOR MODULATOR CONTAINING SAID DERIVATIVE AS ACTIVE INGREDIENT Russian patent published in 2011 - IPC C07F9/09 A61K31/661 A61P9/10 

Abstract RU 2430925 C2

FIELD: chemistry.

SUBSTANCE: invention relates to aminophosphate derivatives of general formula (1a), pharmaceutically acceptable salts or hydrates thereof, which can be used in medicine as S1P (sphingosine-1-phosphate) receptor modulators,

where R3 is a straight alkyl group containing 1-3 carbon atoms; X is an oxygen or sulphur atom and n equals 2 or 3.

EFFECT: obtaining novel biologically active compounds with high S1P receptor modulating action.

9 cl, 59 ex, 1 tbl

Similar patents RU2430925C2

Title Year Author Number
AMINO ALCOHOL AND IMMUNODEPRESSANT CONTAINING IT AS ACTIVE INGREDIENT 2007
  • Kokhno Jasushi
  • Fudzhii Kijoshi
  • Saito Tatsukhiro
  • Kurijama Kazukhiko
  • Jasue Tokutarou
RU2458044C2
CYCLOPENTYLACRYLAMIDE DERIVATIVE 2009
  • Fukuda Jasumichi
  • Asakhina Joshikazu
  • Takadoi Masanori
  • Jamamoto Masanori
RU2565070C2
COMPOUNDS USEFUL AS TRPM8 MODULATORS 2011
  • Prist Chad
  • Nonkovich Alen
  • Petron Endryu
  • Ung Dzhejn
RU2608109C2
BIPHENYL DERIVATIVES AND PHARMACEUTICAL AND COSMETIC COMPOSITIONS COMPRISING THEREOF 1998
  • Bernardon Zhan-Mishel'
  • Nedonsel' Filipp
RU2193552C2
QUINOLINE DERIVATIVES 1995
  • Jutaka Nomura
  • Sogo Sakuma
  • Seiitiro Masui
RU2137770C1
AMINO ALCOHOL DERIVATIVES 2005
  • Khattori Koudzi
  • Toda Susumu
  • Vasizuka Keniti
  • Ito Sindzi
  • Tanabe Daisuke
  • Araki Takanobu
  • Sakurai Minoru
RU2399614C2
AZADECALINS CONDENSED WITH HETEROARYLKETONES - GLUCOCORTICOID RECEPTOR MODULATORS 2013
  • Khant Khejzel
  • Dzhonson Toni
  • Rej Nikolas
  • Uolters Ajejn
RU2639867C2
METHOD FOR REDUCING OF BROKEN OPYOID RECEPTOR FUNCTIONS 1996
  • Roberts Ehdvard
  • Plobek Niklas
  • Valestedt Klaes
RU2307833C2
DERIVATIVES OF PIPERAZINE AND PIPERIDINE AND PHARMACEUTICAL COMPOSITION 1996
  • Roberts Ehdvard
  • Plobek Niklas
  • Valestedt Klaes
RU2194702C2
FIVE-MEMBERED HETEROCYCLIC PYRIDINE COMPOUNDS AND PREPARATION METHOD AND USE THEREOF 2014
  • Shen Tszinkan
  • Gen Mejyuj
  • Din Tszyan
  • Syu Bin
  • Aj Tszin
  • Ma Yujchi
  • Van Syu
  • Pen Sya
  • Chen Yuelej
  • Chen Dantsi
  • Men Tao
  • Ma Lanpin
  • Tszi Inchun
RU2668074C2

RU 2 430 925 C2

Authors

Kokhno Jasushi

Fudzhii Kijoshi

Saito Tatsukhiro

Dates

2011-10-10Published

2007-08-07Filed