AMINOPHOSPHATE DERIVATIVE AND S1P RECEPTOR MODULATOR CONTAINING SAID DERIVATIVE AS ACTIVE INGREDIENT Russian patent published in 2011 - IPC C07F9/09 A61K31/661 A61P9/10 

Abstract RU 2430925 C2

FIELD: chemistry.

SUBSTANCE: invention relates to aminophosphate derivatives of general formula (1a), pharmaceutically acceptable salts or hydrates thereof, which can be used in medicine as S1P (sphingosine-1-phosphate) receptor modulators,

where R3 is a straight alkyl group containing 1-3 carbon atoms; X is an oxygen or sulphur atom and n equals 2 or 3.

EFFECT: obtaining novel biologically active compounds with high S1P receptor modulating action.

9 cl, 59 ex, 1 tbl

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RU 2 430 925 C2

Authors

Kokhno Jasushi

Fudzhii Kijoshi

Saito Tatsukhiro

Dates

2011-10-10Published

2007-08-07Filed