SYNTHESIS OF ACYLAMINOALKENYLAMIDES, SUITABLE AS ANTAGONISTS OF SUBSTANCE P Russian patent published in 2011 - IPC C07D223/12 A61K31/55 A61P1/00 A61P11/00 

Abstract RU 2433122 C2

FIELD: medicine, pharmaceutics.

SUBSTANCE: in claimed invention described is method of obtaining compounds of formula (I) by interaction of compound with base and following interaction of formed compound with compound , where R, R1, R2, R3, R5, T and X have values, given in invention formula.

EFFECT: compounds of formula I are suitable for treatment of a number of conditions, related with substance P and neurokinin.

5 cl, 1 ex

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RU 2 433 122 C2

Authors

Portmann Robert

Dates

2011-11-10Published

2007-04-11Filed