(1-AZABICYCLO[3,3,1]NON-4-YL)-[5-(1H-INDOL-5-YL)-HETEROARYL]-AMINES AS CHOLINERGIC LIGANDS nChAR FOR TREATING PSYCHOTIC AND NEURODEGENERATIVE DISORDERS Russian patent published in 2012 - IPC C07D471/08 A61K31/439 A61P25/00 

Abstract RU 2440350 C2

FIELD: chemistry.

SUBSTANCE: invention describes a compound of formula (III) in form of a free base or an acid addition salt, use thereof as a pharmaceutical agent for preventing, treating and/or inhibiting progression of psychotic and neurodegenerative disorders, as well as pharmaceutical compositions based on said compound.

EFFECT: novel compound which can be used to prevent, treat or inhibit progression of diseases or a pathologic condition in which nAChR α7 activation participates or plays a role.

8 cl, 2 ex

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RU 2 440 350 C2

Authors

Frederiksen Matias

Fojerbakh Dominik

Khurt Konstantse

Koller Manuehl'

Roj Bernar Ljus'En

Dates

2012-01-20Published

2006-12-14Filed