FIELD: pharmacology.
SUBSTANCE: invention refers to the area of chemistry, chemical and pharmaceutical industry and medicine and refers to compounds of formula (1) that can be useful as antipsychotic drugs. Described compounds of formula (1) are the derivatives of 5H-dibenzo[b, e][1, 4]diazepine or its pharmacologically acceptable salts with acid and application of the compounds. Compounds of formula (1) possess higher activity compared to clozapine.
EFFECT: improved antipsychotic effect.
8 cl, 23 ex, 2 tbl
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Authors
Dates
2012-02-10—Published
2010-05-13—Filed