NEW COMPOUNDS ACTING AS ERK INACTIVATORS Russian patent published in 2012 - IPC C07D231/56 C07D403/12 C07D409/12 C07D413/12 C07D417/12 A61K31/506 A61K31/427 A61K31/428 A61K31/496 A61P35/00 C07D417/14 C07D403/14 

Abstract RU 2442778 C9

FIELD: chemistry.

SUBSTANCE: invention refers to new indazole derivants with the formula (1.0) or to their pharmaceutically acceptable salts and isomerides that act as inactivators in relation to ERK2. In formula (1.0): meanings of the chemical groups Q, R1, R2 are given in the invention formula. The invention also refers to the pharmaceutical composition containing the mentioned compounds and to application of the compounds with the formula (1.0) for production of crude drugs used in malignant growth treatment.

EFFECT: application of the compounds for production of crude drugs used in malignant growth treatment.

65 cl, 611 ex, 27 tbl

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RU 2 442 778 C9

Authors

Kuper Alan

Deng Jongki

Shipps Dzheral'D V. Ml.

Shikh Neng-Jang

Zhu Kh'Ju

San Robert

Kelli Dzhozef

Doll Ronal'D

Nan Jang

Vang Tong

Desai Jagdish

Vang Dzhejms

Dong Jukhao

Mehdison Vinsent S.

Ksiao Li

Khruza Alan

Siddiki M. Arshad

Samatar Akhmed

Palival Sunil

Tsui Khon-Chung

Chelebi Azim A.

Vu Jidzhi

Boga Sobkhana Babu

Dates

2012-02-20Published

2006-12-11Filed