METHOD OF PRODUCING 5,6-DIHYDRO-7H-PYRROLO[1,2-d][1,4]BENZODIAZEPIN-6-ONE DERIVATIVES Russian patent published in 2012 - IPC C07D243/06 C07D487/04 A61K31/5517 

Abstract RU 2455289 C1

FIELD: chemistry.

SUBSTANCE: invention relates to organic chemistry and synthesis of heterocyclic compounds - 5,6-dihydro-7H-pyrrolo[1,2-d][1,4]benzodiazepin-6-one derivatives of formula 1a-e by boiling 2-amino-N-(2-furan-2-yl-phenyl)-acetamides in a mixture of glacial acetic acid and concentrated hydrochloric acid with subsequent treatment with sodium bicarbonate while boiling.

EFFECT: method is characterised by simple execution.

2 tbl, 5 ex

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RU 2 455 289 C1

Authors

Shcherbinin Vitalij Aleksandrovich

Nevolina Tat'Jana Nikolaevna

Butin Aleksandr Valerianovich

Dates

2012-07-10Published

2011-05-05Filed