FIELD: chemistry.
SUBSTANCE: invention relates to organic chemistry and synthesis of heterocyclic compounds - 5,6-dihydro-7H-pyrrolo[1,2-d][1,4]benzodiazepin-6-one derivatives of formula 1a-e by boiling 2-amino-N-(2-furan-2-yl-phenyl)-acetamides in a mixture of glacial acetic acid and concentrated hydrochloric acid with subsequent treatment with sodium bicarbonate while boiling.
EFFECT: method is characterised by simple execution.
2 tbl, 5 ex
Title | Year | Author | Number |
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METHOD OF PRODUCING 5,6-DIHYDRO-4H-BENZO[f]PYRROLO[1,2-α][1,4]DIAZEPIN-6-ONE | 2010 |
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RU2425037C1 |
METHOD OF PRODUCING 1,2-DIHYDROPYRROLO[1,2-a]PYRAZIN-3(4H)-ONE DERIVATIVES | 2012 |
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RU2490271C1 |
METHOD FOR PREPARATION OF DERIVATIVES OF PYRROLO[1,2-a][1,4]DIAZEPINE | 2006 |
|
RU2323939C1 |
METHOD FOR SYNTHESIS OF 10-METHYL-6,7-DIHYDRO-5H-PYRROLO[1,2-a][1,5]BENZODIAZEPINE DERIVATIVES | 2015 |
|
RU2603344C1 |
METHOD OF OBTAINING DERIVATIVES OF 2-DIALKYLAMINOPYRROLO[1,2-ALPHA][1,4]BENZODIAZEPINE | 2012 |
|
RU2518102C1 |
METHOD FOR PRODUCING OF 7-ALKYL-2,3-DIHYDRO-1H-PYRROLO[1,2-D][1,4]DYAZEPINE-4(5H)-ONE DERIVATIVES | 2017 |
|
RU2659390C1 |
METHOD FOR PREPARING 4-[1-(TOLYL-4-SULFONYL)-1H-INDOLYL-2]-BUT-3-ENE-2-ONE'S | 2005 |
|
RU2294325C2 |
USE OF 1-METHYL-8,9-DIMETHOXY-4,5-DIHYDRO-6H-PYRROLO[1,2-A][1,4]BENZODIAZEPIN-6-ONE AS AN ANTIFUNGAL AGENT AGAINST YEAST FUNGI | 2023 |
|
RU2808993C1 |
HETEROCYCLIC INHIBITORS OF Hh-SYGNAL CASCADE, BASED ON THEM MEDICINAL COMPOSITIONS AND METHOD OF TREATING DISEASES INDUCED BY ABBARANT ACTIVITY OF Hh-SIGNAL SYSTEM | 2007 |
|
RU2364597C1 |
USE OF 1-METHYL-4,5-DIHYDRO-6H-PYRIDO[1,2-a][1,4]BENZODIAZEPINE-6-ONE AS ANTIFUNGAL AGENT AGAINST YEASTS | 2023 |
|
RU2809026C1 |
Authors
Dates
2012-07-10—Published
2011-05-05—Filed