METHOD OF PRODUCING 1,2-DIHYDROPYRROLO[1,2-a]PYRAZIN-3(4H)-ONE DERIVATIVES Russian patent published in 2013 - IPC C07D487/04 

Abstract RU 2490271 C1

FIELD: chemistry.

SUBSTANCE:

which involves recyclisation of a furan ring of 2-amino-N-(furan-2-ymethyl)acetamides at room temperature in a mixture of glacial acetic acid and concentrated hydrochloric acid for 24 hours, after which sodium bicarbonate is added and then boiled for 5 minutes.

EFFECT: novel method of producing 1,2-dihydropyrrolo[1,2-α]pyrazin-3(4H)-ones as a result of simultaneous formation of a pyrrole ring and a pyrazine ring, which in turn can be used as biologically active substances.

1 cl, 3 tbl, 5 ex

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RU 2 490 271 C1

Authors

Shcherbinin Vitalij Aleksandrovich

Nevolina Tat'Jana Anatol'Evna

Shpuntov Pavel Mikhajlovich

Butin Aleksandr Valerianovich

Dates

2013-08-20Published

2012-05-11Filed