BIARYL CARBOXYARYL AMIDES AS TYPE 1 VANILLOID MODULATORS Russian patent published in 2012 - IPC C07D401/04 A61K31/4725 A61P13/00 A61P29/00 

Abstract RU 2468020 C2

FIELD: chemistry.

SUBSTANCE: present invention relates to novel biaryl carboxyaryl amide derivatives of general formula , where: A is N; Z is a phenyl ring substituted with a group R selected from a halogen atom. The invention also relates to use of the compound of formula (I) and to a pharmaceutical composition based on the compound of formula (I).

EFFECT: novel biaryl carboxyaryl amide derivatives, which are useful as type 1 vanilloid receptor modulators, are obtained.

9 cl, 1 ex

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RU 2 468 020 C2

Authors

Baraldi P'Er Dzhovanni

Borea P'Er Andrea

Dzheppetti P'Erandzhelo

Pavani Marija Dzhovanna

Fruttarolo Francheska

Trevizani Marchello

Dates

2012-11-27Published

2007-07-02Filed