FIELD: chemistry.
SUBSTANCE: invention relates to 3-aroyl-2-hydroxy-2-(2-oxocycloalkyl)pyrrolo[2,1-c][1,4]benzoxazine-1,4(2H)-diones of formula (I) , having analgesic activity and a method for production thereof. In general formula (I) Ar = Ph (a-c), C6H4Br-4 (d), C6H4OMe-4 (e), n = 1 (a), 2 (b, d, e), 3 (c).
EFFECT: higher activity of the compounds.
3 cl, 1 tbl, 6 ex
Title |
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Author |
Number |
METHOD FOR PRODUCING (R*)-3-AROYL-2-HYDROXY-2-((S*)-2-OXOCYCLOALKYL)PYRROLO[1,2-A]QUINOXALINE-1,4(2H,5H)-DIONES |
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