(2S,3R-)-N-(2-((3-PYRIDINYL)METHYL)-1-AZABICYCLO[2,2,2]OCT-3-YL)BENZOFURANE-2-CARBOXAMIDE, NEW SALT FORMS AND METHODS FOR PREPARING THEM Russian patent published in 2013 - IPC A61K31/439 A61K31/4545 A61P25/16 

Abstract RU 2476220 C2

FIELD: medicine, pharmaceutics.

SUBSTANCE: present invention refers to organic chemistry and medicine, and concerns salts of (2S,3R-)-N-(2-((3-pyridinyl)methyl)-1-azabicyclo[2.2.2]oct-3-yl)benzofurane-2-carboxamide, substantially free from (2S,3S)-N-(2-((3-pyridinyl)methyl)-1-azabicyclo[2.2.2]oct-3-yl)benzofurane-2-carboxamide, (2R,3S)-N-(2-((3-pyridinyl)methyl)-1-azabicyclo[2.2.2]oct-3-yl)benzofurane-2-carboxamide and (2R,3R)-N-(2-((3-pyridinyl)methyl)-1-azabicyclo[2.2.2]oct-3-yl)benzofurane-2-carboxamide.

EFFECT: preparing the compositions applicable for treating the conditions and disorders associated with central and vegetative nervous system dysfunction.

5 cl, 19 dwg, 7 tbl, 18 ex

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RU 2 476 220 C2

Authors

Bensherif Meruan

Benson Lajza

Dall Gari Moris

Fedorov Nikolaj

Gatto Gregori Dzh.

Dzhenus Dzhon

Dzhordan Kristen G.

Meht'Ju Dzhejkob

Mazurov Anatolij A.

Mjao Lan'

Mun'Os Khulio A.

Pfajffer Inigo

Pfajffer Sondra

Fillips Tereza I.

Dates

2013-02-27Published

2008-08-01Filed