FIELD: medicine, pharmaceutics.
SUBSTANCE: present invention refers to organic chemistry and medicine, and concerns salts of (2S,3R-)-N-(2-((3-pyridinyl)methyl)-1-azabicyclo[2.2.2]oct-3-yl)benzofurane-2-carboxamide, substantially free from (2S,3S)-N-(2-((3-pyridinyl)methyl)-1-azabicyclo[2.2.2]oct-3-yl)benzofurane-2-carboxamide, (2R,3S)-N-(2-((3-pyridinyl)methyl)-1-azabicyclo[2.2.2]oct-3-yl)benzofurane-2-carboxamide and (2R,3R)-N-(2-((3-pyridinyl)methyl)-1-azabicyclo[2.2.2]oct-3-yl)benzofurane-2-carboxamide.
EFFECT: preparing the compositions applicable for treating the conditions and disorders associated with central and vegetative nervous system dysfunction.
5 cl, 19 dwg, 7 tbl, 18 ex
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Authors
Dates
2013-02-27—Published
2008-08-01—Filed