CRYSTALLINE MODIFICATION OF PARA-METHOXYANILIDE OF 6-HYDROXY-4-OXO-2,4-DIHYDRO-1H-PYRROLO[3,2,1-ij]QUINOLINE-5-CARBOXYLIC ACID Russian patent published in 2013 - IPC C07D471/04 A61K31/47 

Abstract RU 2480468 C1

FIELD: chemistry.

SUBSTANCE: invention relates to a novel crystalline modification of para-methoxyanilide of 6-hydroxy-4-oxo-2,4-dihydro-1H-pyrrolo-[3,2,1-ij]quinoline-5-carboxylic acid of formula: (I) , which is obtained by crystallisation from ethyl acetate, where values of interplanar distance (d) and relative reflection intensities (Irel) are given in claim 1.

EFFECT: novel crystalline modification exhibits a high diuretic effect.

2 dwg, 9 tbl, 6 ex

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RU 2 480 468 C1

Authors

Ukrainets Igor' Vasil'Evich

Dates

2013-04-27Published

2012-02-16Filed