4-PYRIMIDINESULPHAMIDE DERIVATIVE Russian patent published in 2013 - IPC C07D403/12 A61K31/506 A61P9/00 A61P25/00 A61P3/10 

Abstract RU 2485116 C2

FIELD: medicine, pharmaceutics.

SUBSTANCE: invention refers to a compound of formula (I) or to a salt thereof: The invention also refers to a method for preparing said compound, a pharmaceutical composition for treating the diseases caused by increased vascular contraction, proliferation or inflammation caused by endothelin on the basis of said compound.

EFFECT: what is prepared is the novel compound and the salts thereof to be used in medicine for treating hypertension, pulmonary hypertension, diabetic arteriopathy, cardiac failure, erectile dysfunction and angina pectoris.

14 cl, 4 tbl, 1 ex

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RU 2 485 116 C2

Authors

Bolli Martin

Boss Kristof

Trajber Aleksander

Dates

2013-06-20Published

2008-08-15Filed