6'-ARYL-2'-(2-HYDROXYPHENYL)-11',11'-DIMETHYL-3',4,4',13'-TETRAOXOSPIRO [2,5-CYCLOHEXADIEN-1,9'-(7'-OXA-2',12'-DIAZATETRACYCLO[6.5.1.0.0]TETRADEC-5'-EN]-14'-CARBOXYLATES AND METHOD FOR PREPARING THEM Russian patent published in 2013 - IPC C07D491/22 A61P29/00 

Abstract RU 2485126 C1

FIELD: medicine, pharmaceutics.

SUBSTANCE: invention refers to 6'-aryl-2'-(2-hydroxyphenyl) - 11',11'-dimethyl- 3', 4, 4', 13'-tetraoxospiro[2,5-cyclohexadien-1,9' - (7' - oxa - 2',12' -diazatetracyclo[6.5.1.01,5.08,2]-tetradec-5'-en]-14'-carboxylates of general formula (IIIa,b) III: Ar=Ph (a), C6H4Me-n (b), and method for preparing them.

EFFECT: preparing the compounds to be used as analgesic agents.

2 cl, 2 ex

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RU 2 485 126 C1

Authors

Konovalova Valerija Vladislavovna

Maslivets Andrej Nikolaevich

Shkljaev Jurij Vladimirovich

Makhmudov Ramiz Ragibovich

Dates

2013-06-20Published

2011-12-29Filed