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(19)

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2 487 866

(13)

(51)

IPC

C07D209/52(2006-01-01)

C07D403/12(2006-01-01)

A61K31/4025(2006-01-01)

(21) (22)

Application

2010128972/04, 2008-05-20

(24)

Start date

2008-05-20

(22)

Actual filing date

2008-05-20

(45)

Published

2013-07-20

(72)

Inventor

Tan Pehn ChzhoLin' ChzhiganLjuj Khehtszjun'Chzhao FutsjanLi LiJan FanlunFu Tszjan'KhunVan LiShehn' Guanjuan'Guan' Dunljan

(73)

Holder

Tszjansu Khehnsokh Farmas'Jutikal Ko., Ltd.Shankhaj Khehnzhuj Farmas'Jutikal Ko., Ltd.

DICYCLOAZAALKANE DERIVATIVES, METHODS FOR PRODUCTION THEREOF AND USE THEREOF IN MEDICINE Russian patent published in 2013 - IPC C07D209/52 C07D403/12 A61K31/4025

Abstract RU 2487866 C2

FIELD: chemistry.

SUBSTANCE: invention relates to azabicycloalkane derivatives of formulae (IB) and (IC) where: R represents the following formula: where values of R, R₁, R₂, R₅-R₇ and W are given in claim 1. The compounds can be used as a dipeptidyl peptidase (DPP-IV) inhibitor.

EFFECT: intermediate compounds and methods of producing compounds IB, IC are described.

22 cl, 1 tbl, 18 ex

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RU 2 487 866 C2

Authors

Tan Pehn Chzho

Lin' Chzhigan

Ljuj Khehtszjun'

Chzhao Futsjan

Li Li

Jan Fanlun

Fu Tszjan'Khun

Van Li

Shehn' Guanjuan'

Guan' Dunljan

Dates

2013-07-20—Published

2008-05-20—Filed