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IPC

C07D207/10(2006-01-01)

A61K31/395(2006-01-01)

A61P23/02(2006-01-01)

(21) (22)

Application

2012115376/15, 2012-04-17

(24)

Start date

2012-04-17

(22)

Actual filing date

2012-04-17

(45)

Published

2014-01-20

(72)

Inventor

Kalinin Dmitrij VadimovichPantsurkin Vladimir IvanovichSyropjatov Boris JakovlevichVakhrin Mikhail Ivanovich

(73)

Holder

Gosudarstvennoe Bjudzhetnoe Obrazovatel'Noe Uchrezhdenie Vysshego Professional'Nogo Obrazovanija Gosudarstvennaja Farmatsevticheskaja Akademija" Ministerstva Zdravookhranenija I Sotsial'Nogo Razvitija Rossijskoj Federatsii Vpo Pgfa Minzdravsotsrazvitija Rossii)

2,6-DIMETHYLANILIDE OF N-CYCLOHEXYLPYRROLIDINE-2-CARBOXYLIC ACID HYDROCHLORIDE, HAVING SURFACE, INFILTRATION AND CONDUCTION ANAESTHESIA ACTIVITY Russian patent published in 2014 - IPC C07D207/10 A61K31/395 A61P23/02

Abstract RU 2504538 C2

FIELD: chemistry.

SUBSTANCE: invention relates to a novel biologically active 2,6-dimethylanilide of N-cyclohexylpyrrolidine-2-carboxylic acid, having surface, infiltration and conduction anaesthesia activity, considerably better than bupivacaine and ropivacaine with the same or less toxicity.

EFFECT: improved compounds.

2 tbl

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RU 2 504 538 C2

Authors

Kalinin Dmitrij Vadimovich

Pantsurkin Vladimir Ivanovich

Syropjatov Boris Jakovlevich

Vakhrin Mikhail Ivanovich

Dates

2014-01-20—Published

2012-04-17—Filed