FIELD: medicine, pharmaceutics.
SUBSTANCE: invention relates to novel compounds of formula
,
where values A, R1-R6 are given in i.1 of the invention formula. Methods of obtaining the formula (I) compound are described.
EFFECT: compounds demonstrate an inhibiting activity of the cathepsin enzyme, which makes it possible to use them for the preparation of a pharmaceutical composition and for the preparation of a medication.
38 cl, 12 dwg, 495 ex
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Authors
Dates
2014-12-10—Published
2010-04-13—Filed