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(19)

(11)

2 539 565

(13)

(51)

IPC

C07D213/38(2006-01-01)

C07D233/54(2006-01-01)

C07D401/12(2006-01-01)

C07D403/12(2006-01-01)

A61K31/18(2006-01-01)

A61K31/4164(2006-01-01)

A61K51/04(2006-01-01)

A61P35/00(2006-01-01)

C07F13/00(2006-01-01)

(21) (22)

Application

2011127467/04, 2009-12-04

(24)

Start date

2009-12-04

(22)

Actual filing date

2009-12-04

(45)

Published

2015-01-20

(72)

Inventor

Babich Dzhon U.Tsimmerman KrejgDzhojal DzhonMareska Kevin P.Lu GenliangKhil'Er Shon

(73)

Holder

Molik'Jular Insajt Farmas'Jutikalz, Ink.

CA-IX SPECIFIC RADIOPHARMACEUTICAL AGENTS FOR TREATING AND IMAGING MALIGNANT TUMOURS Russian patent published in 2015 - IPC C07D213/38 C07D233/54 C07D401/12 C07D403/12 A61K31/18 A61K31/4164 A61K51/04 A61P35/00 C07F13/00

Abstract RU 2539565 C2

FIELD: medicine, pharmaceutics.

SUBSTANCE: invention refers to compounds of formula I , II or IV , wherein the radical values W, V, R^a, R^b, X, L, R^t, A are presented in the patent claim.

EFFECT: declared compounds identify and bind the CA-IX protein; they can contain a radioactive element for radionuclide imaging or therapeutic application.

27 cl, 1 tbl, 5 dwg, 25 ex

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RU 2 539 565 C2

Authors

Babich Dzhon U.

Tsimmerman Krejg

Dzhojal Dzhon

Mareska Kevin P.

Lu Genliang

Khil'Er Shon

Dates

2015-01-20—Published

2009-12-04—Filed