FIELD: chemistry.
SUBSTANCE: invention relates to method for obtaining derivatives of 2-(2-acylvinyl)indoles I 
by reaction of recyclisation of available 2-tosylaminobenzylfuranes at their successive processing with m-chloroperbenzoic acid, and then by trifluoroacetic acid in dichloromethane.
EFFECT: method makes it possible to stereoselectively obtain target products with high output, as well as to vary substituents in indole core.
2 tbl, 6 ex
| Title | Year | Author | Number |
|---|---|---|---|
| PRODUCTION METHOD OF (E)-4-(INDOL-2-YL)PROP-2-EN-1-ONE DERIVATIVES | 2016 |
|
RU2633999C1 |
| METHOD PRODUCING 4-{1-[(4-METHYLPHENYL)SULPHONYL]-1H-INDOL-2-YL}BUT-3-EN-2-ONE DERIVATIVES | 2012 |
|
RU2488581C1 |
| METHOD OF PRODUCING 2-(2-ACYLVINYL)INDOLES | 2012 |
|
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| METHOD OF OBTAINING DERIVATIVES FROM (E)-2-(2-ACYLVINYL)BENZOFURANE | 2016 |
|
RU2633998C1 |
| METHOD OF PRODUCING 2-(BENZYL)FURAN DERIVATIVES | 2014 |
|
RU2570420C1 |
| METHOD FOR SYNTHESIS OF 4-(1H-INDOL-3-YL)-BUT-3-EN-2-ONE DERIVATIVES | 2009 |
|
RU2409564C1 |
| METHOD OF OBTAINING DERIVATIVES OF 2-ARYL(HETARYL)-1H-INDOLES | 2010 |
|
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| INHIBITORS OF CYTOSOLIC PHOSPHOLIPASE A2 | 2002 |
|
RU2337906C2 |
| METHOD FOR PREPARING 4-[1-(TOLYL-4-SULFONYL)-1H-INDOLYL-2]-BUT-3-ENE-2-ONE'S | 2005 |
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RU2294325C2 |
| INDOLES AS 5-HT MODULATORS | 2007 |
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RU2449990C2 |
