FIELD: chemistry.
SUBSTANCE: invention relates to single-reactor method of Micafungin preparation. Method includes acylation of Micafungin peptide core without isolation of activated side chain of Micafungin and its reaction mixture.
EFFECT: single-reactor method for obtaining makes it possible to reduce synthesis time and increase output.
14 cl, 4 dwg, 1 tbl, 5 ex
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Authors
Dates
2016-02-20—Published
2012-03-26—Filed