COMPOUNDS, COMPOSITIONS AND METHODS SUITABLE FOR CHOLESTEROL MOBILISATION Russian patent published in 2016 - IPC C07D403/14 C07D413/14 C07D401/14 A61K31/506 A61K31/5377 A61K31/4427 A61P3/00 

FIELD: chemistry.

SUBSTANCE: invention relates to organic chemistry, specifically to a novel heterocyclic compound of general formula (II) or to a pharmaceutically acceptable salt, where each R⁹ is -H; each R¹⁰ is independently -H, -OH, NH(methyl), -N(methyl)(methyl) or -O-methyl; each of Q¹, Q² and Q³ is independently CR¹⁰ or N; X is CHR¹⁰ or O; and each m is 1. The invention also relates to a pharmaceutical composition based on a compound of formula (II), a treatment method based on the use of a compound of formula (II), and a method of determining the level of activity of P2Y13 in a subject, based on the use of a compound of formula (II).

EFFECT: obtaining novel compounds having agonistic activity with respect to the P2Y13 receptor.

18 cl, 28 dwg, 4 tbl, 20 ex